Efficient TCT-catalyzed synthesis of 1,5-benzodiazepine derivatives under mild conditions.
نویسندگان
چکیده
2,4,6-Trichloro-1,3,5-triazine (TCT) efficiently catalyzed the condensation reactions between 1,2-diamines and various enolizable ketones to afford 1,5-benzodiazepines in good to excellent yields. Simple and mild reaction conditions, the use of a cheap catalyst and easy workup and isolation are notable features of this method.
منابع مشابه
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ورودعنوان ژورنال:
- Molecules
دوره 13 9 شماره
صفحات -
تاریخ انتشار 2008